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Research Use Only — Not for Human Consumption

PT-141 (Bremelanotide)

PT-141, also known as Bremelanotide, is a synthetic cyclic heptapeptide and melanocortin receptor agonist. It is structurally derived from Melanotan II (MT-2) but differs in that the C-terminal amide is replaced with a hydroxyl group, making it non-cyclic at the C-terminus while retaining the core cyclic disulfide structure. PT-141 acts as an agonist at melanocortin receptor subtypes (particularly MC1R, MC3R, MC4R, and MC5R). Heartland Bio Labs supplies PT-141 as a lyophilized research compound of verified purity.

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PT-141, also known by the name bremelanotide in the research literature, is a synthetic cyclic heptapeptide agonist of the melanocortin receptor family, with particular activity at the MC3 and MC4 receptors. It was developed from the melanocortin analogue Melanotan II, and it occupies a distinctive place in peptide research: most compounds in this catalog act on metabolic, repair, or neurotrophic pathways, while PT-141 is the catalog's window into central melanocortin signaling. Heartland Bio Labs supplies PT-141 for laboratory research in 10mg vials with independent verification.

What PT-141 is

PT-141 descends directly from Melanotan 2, and the structural change between them is what shifted the research focus. Our Melanotan 2 vs PT-141 comparison covers the lineage and the differences that matter.

The melanocortin system is a signaling network built around alpha-MSH and its receptors, MC1 through MC5, governing a wide range of processes studied across pigmentation, energy balance, inflammation, and central nervous system research. PT-141 is a cyclized, modified analogue in that family: the ring structure gives it stability the linear parent lacks, and its receptor profile concentrates on MC3R and MC4R, the receptors most studied in central signaling research. Structural background is in our PT-141 research overview.

Product characteristics

  • Synthetic cyclic heptapeptide, melanocortin receptor agonist (MC3R/MC4R focus)
  • Derived from the Melanotan II lineage of alpha-MSH analogues
  • Approximate molecular weight: 1,025.2 g/mol
  • Supplied as white lyophilized powder in sealed vials
  • Available strength: 10mg; a 5mg vial appears on the selector with a notify option when not in stock
  • HPLC purity and mass spectrometry identity, tested by an independent laboratory
  • For laboratory research use only

The melanocortin family on this site

PT-141 is not the only melanocortin-derived compound we stock. KPV is the C-terminal tripeptide of alpha-MSH itself, studied on the inflammation-signaling side of the family, and Kisspeptin-10 sits in the adjacent neuroendocrine research space. Laboratories mapping receptor-family signaling often work across these compounds, and each is tested and documented the same way.

How this product is verified

A cyclic peptide is a slightly harder analytical target than a linear one, which makes independent testing more valuable, not less. PT-141 is verified by HPLC for purity and mass spectrometry for identity at an independent laboratory, with certificates published in our COA portal before purchase. Our guide on reading a peptide certificate of analysis explains the document line by line, and the broader checklist lives in how to vet a research peptide supplier.

Pricing, storage, and shipping

The 10mg vial is $85, in stock, shipping same-day from the Tulsa, Oklahoma area on orders placed before 2:00 PM Central. Store lyophilized vials sealed, cool, dry, and away from light, refrigerated for the long term; reconstitute with bacteriostatic water and refrigerate the solution, using it within the window your protocol defines. Institutional quantities run through our wholesale program.

Reconstitution math

Work out concentration (mg/mL), amount per volume and molarity for any vial size with the general peptide calculator. For the bench procedure see how to reconstitute peptides.

Research use only

PT-141 from Heartland Bio Labs is sold strictly for laboratory research and identification purposes. It is not a drug, it has not been evaluated by the FDA, and it is not for human or veterinary use of any kind. By purchasing, you affirm that you are qualified to handle research compounds and agree to our research use policy.

PT-141 has been studied extensively in the context of melanocortin receptor pharmacology, central nervous system melanocortin signaling, and endocrine axis research. It is the subject of a substantial published literature covering MC4R and MC3R agonism, hypothalamic signaling, and behavioral models in rodents and primates. PT-141 has an extensive published reference literature spanning multiple preclinical and translational research models.

This compound is supplied strictly for research purposes. No clinical or therapeutic application is implied or represented.

Analytical specifications for this product are available on request.

For research and laboratory use only. Not for human or veterinary consumption. Not evaluated by the FDA. See full site disclaimer.

Handling Information

Handle PT-141 under standard laboratory conditions with appropriate PPE. Avoid repeated freeze-thaw cycles once reconstituted. This compound is intended for use by qualified research professionals only.

Storage Requirements

  • Long-term (lyophilized): Store at -20°C, protected from light and moisture
  • Short-term (reconstituted): Store at 4°C; use within 14 days
  • Keep in original sealed vial until point of use
How should I store this peptide?+

Lyophilized peptides should be stored at −20°C in a dry, light-protected environment. Avoid repeated freeze-thaw cycles. Once reconstituted, store at 2-8°C and use within 4-8 weeks depending on the compound.

What should I reconstitute it with?+

Bacteriostatic water or sterile water for research use. We recommend our companion BAC Water for consistency. Specific reconstitution volume depends on your research protocol — refer to the Specifications tab for solubility data.

How quickly do orders ship?+

Orders confirmed before 2:00 PM CT ship the same business day from our facility in Tulsa, OK. Standard US transit is 2-5 business days. Tracking provided at shipment.

Is the COA verified independently?+

Yes. Every product is tested by HPLC for purity (target COA-verified purity) and mass spectrometry for molecular identity before release. The COA is generated from the actual test data, not a generic template.

Can I get bulk or institutional pricing?+

Yes — qualified research facilities and high-volume orders receive tiered pricing. Contact us with your institution information and target quantities.

Further reading

View this product's Certificate of Analysis

Every product is independently verified — HPLC purity, mass spec identity, lot number, storage parameters. Click below to view or download.

Look up COA in portal →
Research Use Only: This product is sold by Heartland Bio Labs for research and laboratory use only. Not intended for human or veterinary consumption, administration, or therapeutic use. This product has not been evaluated by the Food and Drug Administration. Not a drug. Not a dietary supplement. Researchers are responsible for compliance with all applicable regulations.